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ECHA InfoCard | 100.222.780 ![]() |
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Formula | C9H13N2O5P |
Molar mass | 260.186 g·mol−1 |
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Perzinfotel (EAA-090) is a drug which acts as a potent NMDA antagonist.[1] It has neuroprotective effects and has been investigated for the treatment of stroke,[2] but lacks analgesic effects.[3] Nevertheless, it shows a good safety profile compared to older drugs, although further development of this drug has been discontinued.[4]
Prodrugs were developed since the oral bioavailability of perzinfotel is only around 3-5%.[5]
AMPARTooltip α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor |
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KARTooltip Kainate receptor |
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NMDARTooltip N-Methyl-D-aspartate receptor |
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